UCL Discovery
UCL home » Library Services » Electronic resources » UCL Discovery

Browse by UCL people

Group by: Type | Date
Jump to: Article
Number of items: 21.

Article

Chetty, S; Armstrong, T; Sharma Kharkwal, S; Drewe, WC; De Matteis, CI; Evangelopoulos, D; Bhakta, S; (2021) New InhA Inhibitors Based on Expanded Triclosan and Di-Triclosan Analogues to Develop a New Treatment for Tuberculosis. Pharmaceuticals , 14 (4) , Article 361. 10.3390/ph14040361. Green open access
file

Danquah, CA; Kakagianni, E; Khondkar, P; Maitra, A; Rahman, M; Evangelopoulos, D; McHugh, TD; ... Gibbons, S; + view all (2018) Analogues of Disulfides from Allium stipitatum Demonstrate Potent Anti-tubercular Activities through Drug Efflux Pump and Biofilm Inhibition. Scientific Reports , 8 , Article 1150. 10.1038/s41598-017-18948-w. Green open access
file

Ferguson, Lindsay; Madieh, Nasrin Shokrzadeh; Vaideanu, Alexandra; Schatzlein, Andreas; Festa, Joseph; Singh, Harprit; Wells, Geoff; ... Brucoli, Federico; + view all (2022) C2-linked alkynyl poly-ethylene glycol(PEG) adenosine conjugates as water-soluble adenosine receptor agonists. Chemical Biology & Drug Design 10.1111/cbdd.14128. (In press). Green open access
file

Ferguson, L; Bhakta, S; Fox, KR; Wells, G; Brucoli, F; (2020) Synthesis and Biological Evaluation of a Novel C8-Pyrrolobenzodiazepine (PBD) Adenosine Conjugate. A Study on the Role of the PBD Ring in the Biological Activity of PBD-Conjugates. Molecules , 25 (5) , Article 1243. 10.3390/molecules25051243. Green open access
file

Ferguson, L; Wells, G; Bhakta, S; Johnson, J; Guzman, J; Parish, T; Prentice, RA; (2019) Integrated target-based and phenotypic screening approaches for the identification of anti-tubercular agents that bind to the mycobacterial adenylating enzyme MbtA. ChemMedChem , 14 (19) pp. 1735-1741. 10.1002/cmdc.201900217. Green open access
file

Guzman, JD; Pesnot, T; Barrera, DA; Davies, HM; McMahon, E; Evangelopoulos, D; Mortazavi, PN; ... Bhakta, S; + view all (2015) Tetrahydroisoquinolines affect the whole-cell phenotype of Mycobacterium tuberculosis by inhibiting the ATP-dependent MurE ligase. J Antimicrob Chemother , 70 (6) pp. 1691-1703. 10.1093/jac/dkv010. Green open access
file

Kerai, LV; Hilton, S; Maugueret, M; Kazi, BB; Faull, J; Bhakta, S; Murdan, S; (2016) UV-curable gels as topical nail medicines:In vivo residence, anti-fungal efficacy and influence of gel components on their properties. International Journal of Pharmaceutics , 514 (1) pp. 244-254. 10.1016/j.ijpharm.2016.08.025. Green open access
file

Maitra, A; Evangelopoulos, D; Chrzastek, A; Martin, LT; Hanrath, A; Chapman, E; Hailes, HC; ... Bhakta, S; + view all (2020) Carprofen elicits pleiotropic mechanisms of bactericidal action with the potential to reverse antimicrobial drug resistance in tuberculosis. Journal of Antimicrobial Chemotherapy , Article dkaa307. 10.1093/jac/dkaa307. Green open access
file

Maitra, A; Munshi, T; Healy, J; Martin, LT; Vollmer, W; Keep, NH; Bhakta, S; (2019) Cell wall peptidoglycan in Mycobacterium tuberculosis: An Achilles' heel for the TB-causing pathogen. FEMS Microbiology Reviews , 43 (5) pp. 548-575. 10.1093/femsre/fuz016. Green open access
file

Maitra, A; Nukala, S; Dickman, R; Martin, LT; Munshi, T; Gupta, A; Shepherd, AJ; ... Bhakta, S; + view all (2021) Characterization of the MurT/GatD complex in Mycobacterium tuberculosis towards validating a novel anti-tubercular drug target. JAC-Antimicrobial Resistance , 3 (1) 10.1093/jacamr/dlab028. (In press). Green open access
file

Martin, Liam T; Daniel, Chris; Guldberg-Allen, Marcus; Navaratnarajah, Anushandan; Anselmi, Silvia; Burova, Tina-Maria D; Willcocks, Sam; ... Bhakta, Sanjib; + view all (2025) Development of Carprofen analogues with activity against Mycobacterium tuberculosis. Bioorganic & Medicinal Chemistry , 127 , Article 118226. 10.1016/j.bmc.2025.118226. Green open access
file

Munshi, T; Gupta, A; Evangelopoulos, D; Guzman, JD; Gibbons, S; Keep, NH; Bhakta, S; (2013) Characterisation of ATP-Dependent Mur Ligases Involved in the Biogenesis of Cell Wall Peptidoglycan in Mycobacterium tuberculosis. PLoS One , 8 (3) , Article e60143. 10.1371/journal.pone.0060143. Green open access
file

Osman, K; Evangelopoulos, D; Basavannacharya, C; Gupta, A; McHugh, TD; Bhakta, S; Gibbons, S; (2012) An antibacterial from Hypericum acmosepalum inhibits ATP-dependent MurE ligase from Mycobacterium tuberculosis. International Journal of Antimicrobial Agents , 39 (2) 124 - 129. 10.1016/j.ijantimicag.2011.09.018. Green open access
file

Quay, DHX; Cole, AR; Cryar, A; Thalassinos, K; Williams, MA; Bhakta, S; Keep, NH; (2015) Structure of the stationary phase survival protein YuiC from B.subtilis. BMC Structural Biology , 15 , Article 12. 10.1186/s12900-015-0039-z. Green open access
file

Rizi, K; Xu, K; Begum, T; Faull, J; Bhakta, S; Murdan, S; (2022) A drug-in-adhesive anti-onychomycotic nail patch: Influence of drug and adhesive nature on drug release, ungual permeation, in vivo residence in human and anti-fungal efficacy. International Journal of Pharmaceutics , 614 , Article 121437. 10.1016/j.ijpharm.2021.121437. Green open access
file

Rizi, K; Murdan, S; Danquah, CA; Faull, J; Bhakta, S; (2015) Development of a rapid, reliable and quantitative method: "SPOTi" for testing antifungal efficacy. Journal of Microbiological Methods , 117 pp. 36-40. 10.1016/j.mimet.2015.07.005. Green open access
file

Ryan, A; Polycarpou, E; Lack, NA; Evangelopoulos, D; Sieg, C; Halman, A; Bhakta, S; ... Sim, E; + view all (2017) Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. British Journal of Pharmacology , 174 (14) pp. 2209-2224. 10.1111/bph.13810. Green open access
file

Shyam, M; Verma, H; Bhattacharje, G; Mukherjee, P; Singh, S; Kamilya, S; Jalani, P; ... Jayaprakash, V; + view all (2022) Mycobactin Analogues with Excellent Pharmacokinetic Profile Demonstrate Potent Antitubercular Specific Activity and Exceptional Efflux Pump Inhibition. Journal of Medicinal Chemistry , 65 (1) pp. 234-256. 10.1021/acs.jmedchem.1c01349. Green open access
file

Teo, SP; Bhakta, S; Stapleton, P; Gibbons, S; (2020) Bioactive Compounds from the Bornean Endemic Plant Goniothalamus longistipetes. Antibiotics , 9 (12) , Article 913. 10.3390/antibiotics9120913. Green open access
file

Touitou, M; Manetti, F; Ribeiro, CM; Pavan, FR; Scalacci, N; Zrebna, K; Begum, N; ... Castagnolo, D; + view all (2020) Improving the Potency of N-Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria. ACS Medicinal Chemistry Letters , 11 (5) pp. 638-644. 10.1021/acsmedchemlett.9b00515. Green open access
file

Xia, DQH; Qureshi, A; Bhakta, S; Keep, NH; (2018) Mutation studies of the gene encoding YuiC, a stationary phase survival protein in Bacillus subtilis. Malaysian Journal of Microbiology , 14 (6) pp. 444-451. 10.21161/mjm.1461801. Green open access
file

This list was generated on Sun Feb 8 05:07:46 2026 GMT.