Browse by UCL people
Group by: Type | Date
Number of items: 18.
Article
AlKharboush, DF;
Kozielski, F;
Wells, G;
Porta, EOJ;
(2025)
Fragment-based drug discovery: A graphical review.
Current Research in Pharmacology and Drug Discovery
, 9
, Article 100233. 10.1016/j.crphar.2025.100233.
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Ballari, MS;
O. J. Porta, E;
Zalazar, EA;
Etichetti, CMB;
Padrón, JM;
Girardini, JE;
Labadie, GR;
(2023)
Lipophilic modification of salirasib modulates the antiproliferative and antimigratory activity.
Bioorganic and Medicinal Chemistry
, 92
, Article 117417. 10.1016/j.bmc.2023.117417.
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Charlton, Rebecca;
Escrivani, Douglas;
Brown, Christopher;
Thota, Niranjan;
de Sousa Agostino, Victor;
Porta, Exequiel;
Avkiran, Timur;
... Steel, PG; + view all
(2025)
Simple Accessible Clemastine Fumarate Analogues as Effective Antileishmanials.
RSC Medicinal Chemistry
10.1039/D4MD01004C.
(In press).
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Díaz-Storani, L;
Clary, AA;
Moreno, DM;
Ballari, MS;
Porta, EOJ;
Bracca, ABJ;
Johnston, JB;
(2021)
Synthesis and interaction of terminal unsaturated chemical probes with Mycobacterium tuberculosis CYP124A1.
Bioorganic and Medicinal Chemistry
, 44
, Article 116304. 10.1016/j.bmc.2021.116304.
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Isern, Jaime A;
Carlucci, Renzo;
Labadie, Guillermo R;
Porta, Exequiel OJ;
(2025)
Progress and Prospects of Triazoles in Advanced Therapies for Parasitic Diseases.
Tropical Medicine and Infectious Disease
, 10
(5)
, Article 142. 10.3390/tropicalmed10050142.
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Isern, Jaime A;
Porta, Exequiel OJ;
Kalesh, Karunakaran;
Koutsogiannis, Zisis;
Cazzola, Davide;
Pohl, Ehmke;
Denny, Paul;
(2025)
Profiling Serine Hydrolases in the Leishmania Host‐Pathogen Interactome Using Cell‐Permeable Activity‐Based Fluorophosphonate Probes.
ChemBioChem
10.1002/cbic.202500160.
(In press).
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Milian, Julieta Litka;
Duché, Geneviève;
Porta, Exequiel;
Harvey-Reid, Alexander;
Clough, Sophie;
Shearman, Billie;
Bedwell, Elizabeth;
(2025)
Amplifying Student Voices in Curriculum Decolonisation: A Collaborative Journey in Higher Education Chemistry.
Student Engagement in Higher Education Journal
, 7
(1)
pp. 20-38.
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Mina, JG;
Parthasarathy, A;
Porta, EO;
Denny, PW;
Kalesh, K;
(2024)
BONCAT-iTRAQ Labelling Reveals Molecular Markers of Adaptive Responses in Toxoplasma gondii to Pyrimethamine Treatment.
Pathogens
, 13
(10)
, Article 879. 10.3390/pathogens13100879.
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Porta, EO;
Gao, L;
Denny, PW;
Steel, PG;
Kalesh, K;
(2023)
Inhibition of HSP90 distinctively modulates the global phosphoproteome of Leishmania mexicana developmental stages.
Microbiology Spectrum
, 11
(6)
, Article e0296023. 10.1128/spectrum.02960-23.
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Porta, EOJ;
(2023)
Mapping the Evolution of Activity-Based Protein Profiling: A Bibliometric Review.
Advanced Pharmaceutical Bulletin
, 13
(4)
pp. 639-645.
10.34172/apb.2023.082.
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Porta, EOJ;
Ballari, MS;
Carlucci, R;
Wilkinson, S;
Ma, G;
Tekwani, BL;
Labadie, GR;
(2023)
Systematic study of 1,2,3-triazolyl sterols for the development of new drugs against parasitic Neglected Tropical Diseases.
European Journal of Medicinal Chemistry
, 254
, Article 115378. 10.1016/j.ejmech.2023.115378.
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Porta, EOJ;
Isern, JA;
Kalesh, K;
Steel, PG;
(2022)
Discovery of Leishmania Druggable Serine Proteases by Activity-Based Protein Profiling.
Frontiers in Pharmacology
, 13
, Article 929493. 10.3389/fphar.2022.929493.
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Porta, EOJ;
Kalesh, K;
Isern, JA;
Steel, PG;
(2025)
Microplate-Based Enzymatic Activity Assay Protocol Powered by Activity-Based Probes.
Methods in Molecular Biology
, 2921
pp. 119-137.
10.1007/978-1-0716-4502-4_6.
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Porta, EOJ;
Kalesh, K;
Steel, PG;
(2023)
Navigating drug repurposing for Chagas disease: advances, challenges, and opportunities.
Frontiers in Pharmacology
, 14
, Article 1233253. 10.3389/fphar.2023.1233253.
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Porta, EOJ;
Steel, PG;
(2023)
Activity-based protein profiling: A graphical review.
Current Research in Pharmacology and Drug Discovery
, 5
, Article 100164. 10.1016/j.crphar.2023.100164.
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Porta, Exequiel OJ;
(2024)
The crucial role of drug repositioning in tackling Chagas disease, sleeping sickness, and leishmaniasis.
INNOSC Theranostics and Pharmacological Sciences
, 7
(4)
, Article 3721. 10.36922/itps.3721.
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Porta, Exequiel OJ;
Saffaei, Ali;
Kalesh, Karunakaran;
(2024)
Editorial: The evolution in pharmacology of infectious diseases: 2022.
Frontiers in Pharmacology
, 15
, Article 1386077. 10.3389/fphar.2024.1386077.
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Book
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Porta, Exequiel and Saffaei, Ali and Kalesh, Karunakaran (Eds).
(2024)
The Evolution in Pharmacology of Infectious Diseases: 2022.
[Book].
Frontiers Media SA: Lausanne, Switzerland.
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