Browse by UCL people
Group by: Type | Date
Number of items: 13.
Article
Dines, JA;
Marson, CM;
(2016)
A direct alkylation route to branched derivatives of suberoylanilide hydroxamic acid (SAHA), a potent non-selective inhibitor of histone deacetylases.
Tetrahedron
, 72
(52)
pp. 8584-8592.
10.1016/j.tet.2016.11.039.
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Greenwood, SOR;
Chan, AWE;
Hansen, DF;
Marson, CM;
(2020)
Potent non-hydroxamate inhibitors of histone deacetylase-8: Role and scope of an isoindolin-2-yl linker with an α-amino amide as the zinc-binding unit.
Bioorganic & Medicinal Chemistry Letters
, 30
(5)
, Article 126926. 10.1016/j.bmcl.2019.126926.
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Marson, C;
Waugh, T;
Masters, J;
Aliev, A;
(2020)
Monocyclic Quinone Structure-Activity Patterns: Synthesis of Catalytic Inhibitors of Topoisomerase II with Potent Anti-Proliferative Activity.
ChemMedChem
, 15
(1)
pp. 114-124.
10.1002/cmdc.201900548.
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Marson, CM;
Koo, CY;
Reyes-Corral, M;
Olmos, Y;
Tavares, IA;
Linardopoulos, S;
Tutt, A;
(2017)
Targeting TAO kinases using a new inhibitor compound delays mitosis and induces mitotic cell death in centrosome amplified breast cells.
Molecular Cancer Therapeutics
, 16
(11)
pp. 2410-2421.
10.1158/1535-7163.MCT-17-0077.
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Marson, CM;
Matthews, CJ;
Atkinson, SJ;
Lamadema, N;
Thomas, NS;
(2015)
Potent and selective inhibitors of histone deacetylase-3 containing chiral oxazoline capping groups and a N-(2-Aminophenyl)-benzamide binding unit.
Journal of Medicinal Chemistry
, 58
(17)
pp. 6803-6818.
10.1021/acs.jmedchem.5b00545.
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Marson, CM;
Yau, KC;
(2015)
Regioselective synthesis of substituted piperidine-2,4-diones and their derivatives via Dieckmann cyclisations.
Tetrahedron
, 71
(39)
pp. 7459-7469.
10.1016/j.tet.2015.06.052.
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McCarthy, S;
Marson, CM;
(2022)
A stepwise lactol carbocyclisation to bridged ethers via a keto–acetal cascade.
Journal of Chemical Research
, 46
(1)
pp. 1-8.
10.1177/17475198221079498.
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Pontiki, E;
Hadjipavlou-Litina, D;
Patsilinakos, A;
Tran, TM;
Marson, CM;
(2015)
Pteridine-2,4-diamine derivatives as radical scavengers and inhibitors of lipoxygenase that can possess anti-inflammatory properties.
Future Medicinal Chemistry
, 7
(14)
pp. 1937-1951.
10.4155/fmc.15.104.
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Promontorio, R;
Richard, J-A;
Marson, CM;
(2018)
Late-stage fluorination of bridged scaffolds: chemoselective generation of a CHF group at three positions of the bicyclo[3.3.1]nonane system.
Tetrahedron Letters
, 59
(13)
pp. 1226-1229.
10.1016/j.tetlet.2018.02.038.
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Promontorio, R;
Richard, J-A;
Marson, CM;
(2016)
Domino Michael-aldol annulations for the stereocontrolled synthesis of bicyclo[3.3.1]nonane and bicyclo[3.2.1]octane derivatives.
RSC Advances
, 6
(115)
pp. 114412-114424.
10.1039/C6RA23523A.
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Werbeck, ND;
Shukla, VK;
Kunze, MBA;
Yalinca, H;
Pritchard, RB;
Siemons, L;
Mondal, S;
... Hansen, DF; + view all
(2020)
A distal regulatory region of a class I human histone deacetylase.
Nature Communications
, 11
(1)
, Article 3841. 10.1038/s41467-020-17610-w.
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Thesis
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Greenwood, SOR;
(2016)
Design and evaluation of novel histone deacetylase 8 inhibitors.
Doctoral thesis , UCL (University College London).
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Matthews, CJ;
(2016)
Histone deacetylase inhibitors containing chiral heterocyclic capping groups.
Doctoral thesis , UCL (University College London).
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