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Number of items: 68.
A
Agapouda, A;
Booker, A;
Kiss, T;
Hohmann, J;
Heinrich, M;
Csupor, D;
(2019)
Quality control of Hypericum perforatum L. analytical challenges and recent progress.
Journal of Pharmacy and Pharmacology
, 71
(1)
pp. 15-37.
10.1111/jphp.12711.
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Allardyce, Duncan J;
Bell, Celia M;
Loizidou, Eriketi Z;
(2019)
Argyrin B, a non-competitive inhibitor of the human immunoproteasome exhibiting preference for β1i.
Chemical Biology & Drug Design
, 94
(2)
pp. 1556-1579.
10.1111/cbdd.13539.
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Allen, BDW;
Hareram, MD;
Seastram, AC;
McBride, T;
Wirth, T;
Browne, DL;
Morrill, LC;
(2019)
Manganese-Catalyzed Electrochemical Deconstructive Chlorination of Cycloalkanols via Alkoxy Radicals.
Organic Letters
, 21
(22)
pp. 9241-9246.
10.1021/acs.orglett.9b03652.
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Allocco, AA;
Jin, SC;
Duy, PQ;
Furey, CG;
Zeng, X;
Dong, W;
Nelson-Williams, C;
... Kahle, KT; + view all
(2019)
Recessive Inheritance of Congenital Hydrocephalus With Other Structural Brain Abnormalities Caused by Compound Heterozygous Mutations in ATP1A3.
Frontiers in Cellular Neuroscience
, 13
, Article 425. 10.3389/fncel.2019.00425.
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Asquith, C;
Laitinen, T;
Konstantinova, L;
Tizzard, G;
Poso, A;
Rakitin, O;
Hofmann-Lehmann, R;
(2019)
Investigation of the Pentathiepin Functionality as an Inhibitor of Feline Immunodeficiency Virus (FIV) via a Potential Zinc Ejection Mechanism, as a Model for HIV Infection.
ChemMedChem
, 14
(4)
pp. 454-461.
10.1002/cmdc.201800718.
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Asquith, CRM;
Konstantinova, LS;
Tizzard, GJ;
Laitinen, T;
Coles, SJ;
Rakitin, OA;
Hilton, ST;
(2019)
Exploration and Development of a C–H-Activated Route to Access the [1,2]Dithiolo[4,3-b]indole-3(4H)-thione Core and Related Derivatives.
Synlett
, 30
(2)
pp. 156-160.
10.1055/s-0037-1611692.
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Asquith, CRM;
Sil, BC;
Laitinen, T;
Tizzard, GJ;
Coles, SJ;
Poso, A;
Hofmann-Lehmann, R;
(2019)
Novel epidithiodiketopiperazines as anti-viral zinc ejectors of the Feline Immunodeficiency Virus (FIV) nucleocapsid protein as a model for HIV infection.
Bioorganic & Medicinal Chemistry
, 27
(18)
pp. 4174-4184.
10.1016/j.bmc.2019.07.047.
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B
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Bhamra, SK;
Slater, A;
Howard, C;
Heinrich, M;
Johnson, MRD;
(2019)
Health care professionals' personal and professional views of herbal medicines in the United Kingdom.
Phytotherapy Research
, 33
(9)
pp. 2360-2368.
10.1002/ptr.6418.
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Booker, A;
Chatzinasiou, L;
Heinrich, M;
MacLennan, E;
Mackonochie, M;
(2019)
Turmeric (Curcuma longa L.) products: What quality differences exist?
Journal of Herbal Medicine
, 17-18
, Article 100281. 10.1016/j.hermed.2019.100281.
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Breen, A;
Wells, G;
Turyanska, L;
Bradshaw, T;
(2019)
Development of novel apoferritin formulations for antitumour benzothiazoles.
Cancer Reports
, 2
(4)
, Article e1155. 10.1002/cnr2.1155.
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Breen, AF;
Scurr, D;
Cassioli, ML;
Wells, G;
Thomas, NR;
Zhang, J;
Turyanska, L;
(2019)
Protein Encapsulation of Experimental Anticancer Agents 5F 203 and Phortress: Towards Precision Drug Delivery.
International Journal of Nanomedicine
, 14
pp. 9525-9534.
10.2147/IJN.S226293.
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Brown, P;
Tan, A-C;
El-Esawi, MA;
Liehr, T;
Blanck, O;
Gladue, DP;
Almeida, GMF;
... Shalchyan, V; + view all
(2019)
Large expert-curated database for benchmarking document similarity detection in biomedical literature search.
Database
pp. 1-66.
10.1093/database/baz085.
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Bunc, M;
Hanning, SM;
Prieto Garcia, J;
Kristl, J;
Orlu, M;
(2019)
Characterisation of an in vitro aged cell culture model.
Farmacia
, 67
(2)
pp. 240-247.
10.31925/farmacia.2019.2.7.
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C
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Cao, Q;
Nicholson, WI;
Jones, AC;
Browne, DL;
(2019)
Robust Buchwald-Hartwig amination enabled by ball-milling.
Organic and Biomolecular Chemistry
, 17
(7)
pp. 1722-1726.
10.1039/c8ob01781f.
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Cao, Q;
Stark, RT;
Fallis, IA;
Browne, DL;
(2019)
A Ball-Milling-Enabled Reformatsky Reaction.
ChemSusChem
, 12
(12)
pp. 2554-2557.
10.1002/cssc.201900886.
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Cuadrado, A;
Rojo, A;
Wells, G;
Hayes, J;
Cousin, S;
Rumsey, W;
Attucks, O;
... Dinkova-Kostova, A; + view all
(2019)
Therapeutic targeting of the NRF2 and KEAP1 partnership in chronic diseases.
Nature Reviews Drug Discovery
, 18
pp. 295-317.
10.1038/s41573-018-0008-x.
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D
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Dickman, R;
Danelius, E;
Mitchell, SA;
Hansen, DF;
Erdélyi, M;
Tabor, AB;
(2019)
A Chemical Biology Approach to Understanding Molecular Recognition of Lipid II by Nisin(1-12): Synthesis and NMR Ensemble Analysis of Nisin(1-12) and Analogues.
Chemistry
10.1002/chem.201902814.
(In press).
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Dickman, R;
Mitchell, SA;
Figueiredo, AM;
Hansen, DF;
Tabor, AB;
(2019)
Molecular Recognition of Lipid II by Lantibiotics: Synthesis and Conformational Studies of Analogues of Nisin and Mutacin Rings A and B.
The Journal of Organic Chemistry
, 84
(18)
pp. 11493-11512.
10.1021/acs.joc.9b01253.
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Dodoo, CC;
Alomari, M;
Basit, AW;
Stapleton, P;
Gaisford, S;
(2019)
A thermal ink-jet printing approach for evaluating susceptibility of bacteria to antibiotics.
Journal of Microbiological Methods
, Article 105660. 10.1016/j.mimet.2019.105660.
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Dodoo, CC;
Stapleton, P;
Basit, AW;
Gaisford, S;
(2019)
Use of a water-based probiotic to treat common gut pathogens.
International Journal of Pharmaceutics
, 556
pp. 136-141.
10.1016/j.ijpharm.2018.11.075.
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Duran, D;
Zeng, X;
Jin, SC;
Choi, J;
Nelson-Williams, C;
Yatsula, B;
Gaillard, J;
... Kahle, KT; + view all
(2019)
Mutations in Chromatin Modifier and Ephrin Signaling Genes in Vein of Galen Malformation.
Neuron
, 101
10.1016/j.neuron.2018.11.041.
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F
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Ferguson, L;
Wells, G;
Bhakta, S;
Johnson, J;
Guzman, J;
Parish, T;
Prentice, RA;
(2019)
Integrated target-based and phenotypic screening approaches for the identification of anti-tubercular agents that bind to the mycobacterial adenylating enzyme MbtA.
ChemMedChem
, 14
(19)
pp. 1735-1741.
10.1002/cmdc.201900217.
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Frommenwiler, DA;
Booker, A;
Vila, R;
Heinrich, M;
Reich, E;
Cañigueral, S;
(2019)
Comprehensive HPTLC fingerprinting as a tool for a simplified analysis of purity of ginkgo products.
Journal of Ethnopharmacology
, 243
, Article 112084. 10.1016/j.jep.2019.112084.
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G
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Galaverna, R;
Fernandes, LP;
Browne, DL;
Pastre, JC;
(2019)
Continuous flow processing as a tool for the generation of terpene-derived monomer libraries.
Reaction Chemistry & Engineering
, 4
(2)
pp. 362-367.
10.1039/c8re00237a.
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Galaverna, R;
McBride, T;
Pastre, JC;
Browne, DL;
(2019)
Exploring the generation and use of acylketenes with continuous flow processes.
Reaction Chemistry & Engineering
, 4
(9)
pp. 1559-1564.
10.1039/c9re00072k.
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Guneri, D;
Voegeli, R;
Munday, MR;
Rawlings, AV;
(2019)
12R-lipoxygenase activity is reduced in photodamaged facial stratum corneum. A novel activity assay indicates a key function in corneocyte maturation.
International Journal of Cosmetic Science
, 41
(3)
pp. 274-280.
10.1111/ics.12532.
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Guneri, D;
Voegeli, R;
Zhang, C;
Bankousli, A;
Munday, M;
Lane, M;
Rawlings, A;
(2019)
Humidity-dependent ex vivo corneocyte maturation and the importance of transglutaminase and 12R-lipoxygenase activities.
Presented at: Society-for-Investigative-Dermatology (SID) Meeting, Chicago, IL, USA.
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Guneri, D;
Voegeli, R;
Zhang, C;
Bankousli, AL;
Munday, MR;
Rawlings, AV;
(2019)
The importance of 12R-lipoxygenase and transglutaminase activities in the hydration-dependent ex vivo maturation of corneocyte envelopes.
International Journal of Cosmetic Science
, 41
pp. 563-578.
10.1111/ics.12574.
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H
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Heinrich, M;
Hesketh, A;
(2019)
25 years after the 'Rio Convention'––Lessons learned in the context of sustainable development and protecting indigenous and local knowledge.
Phytomedicine
, 53
pp. 332-343.
10.1016/j.phymed.2018.04.061.
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Heinrich, M;
Scotti, F;
Booker, A;
Fitzgerald, M;
Kum, KY;
Löbel, K;
(2019)
Unblocking High-Value Botanical Value Chains: Is There a Role for Blockchain Systems?
Frontiers in Pharmacology
, 10
, Article 396. 10.3389/fphar.2019.00396.
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Hilton, ST;
Kozielski, F;
Penny, M;
Talapatra, S;
(2019)
Design, 3D printing and validation of a novel low-cost high-capacity sitting-drop bridge for protein crystallization.
Journal of Applied Crystallography
, 52
pp. 171-174.
10.1107/S1600576718017545.
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Hobson, NJ;
Weng, X;
Ashford, M;
Thanh, NTK;
Schätzlein, AG;
Uchegbu, IF;
(2019)
Facile aqueous, room temperature preparation of high transverse relaxivity clustered iron oxide nanoparticles.
Colloids and Surfaces A: Physicochemical and Engineering Aspects
, 570
pp. 165-171.
10.1016/j.colsurfa.2019.03.023.
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Hobson, NJ;
Weng, X;
Siow, B;
Veiga, C;
Ashford, M;
Thanh, NT;
Schätzlein, AG;
(2019)
Clustering superparamagnetic iron oxide nanoparticles produces organ-targeted high-contrast magnetic resonance images.
Nanomedicine
, 14
(9)
pp. 1135-1152.
10.2217/nnm-2018-0370.
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I
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Indorato, R-L;
Talapatra, SK;
Lin, F;
Haider, S;
Mackay, SP;
Kozielski, F;
Skoufias, DA;
(2019)
Is the Fate of Clinical Candidate Arry-520 Already Sealed? Predicting Resistance in Eg5–Inhibitor Complexes.
Molecular Cancer Therapeutics
, 18
(12)
pp. 2394-2406.
10.1158/1535-7163.MCT-19-0154.
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K
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Klug, DM;
Diaz-Gonzalez, R;
Pérez-Moreno, G;
Ceballos-Pérez, G;
García-Hernández, R;
Gomez-Pérez, V;
Ruiz-Pérez, LM;
... Pollastri, MP; + view all
(2019)
Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents.
PLoS Neglected Tropical Diseases
, 13
(2)
, Article e0007129. 10.1371/journal.pntd.0007129.
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Kwapong, AA;
Stapleton, P;
Gibbons, S;
(2019)
Inhibiting plasmid mobility: the effect of isothiocyanates on bacterial conjugation.
International Journal of Antimicrobial Agents
, 53
(5)
pp. 629-636.
10.1016/j.ijantimicag.2019.01.011.
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L
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Lane, M;
Sil, B;
Hilton, S;
Hadgraft, J;
Patel, A;
Crowther, J;
Moore, D;
(2019)
A Preliminary Investigation of Additive Manufacture to Fabricate Human Nail Plate Surrogates for Pharmaceutical Testing.
Pharmaceutics
, 11
(6)
, Article 250. 10.3390/pharmaceutics11060250.
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Laudadio, G;
Barmpoutsis, E;
Schotten, C;
Struik, L;
Govaerts, S;
Browne, DL;
Noel, T;
(2019)
Sulfonamide Synthesis through Electrochemical Oxidative Coupling of Amines and Thiols.
Journal of the American Chemical Society (JACS)
, 141
(14)
pp. 5664-5668.
10.1021/jacs.9b02266.
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Lazarou, R;
Heinrich, M;
(2019)
Herbal Medicine: Who Cares? The changing views on medicinal plants and their roles in British lifestyle.
Phytotherapy Research
, 33
(9)
pp. 2409-2420.
10.1002/ptr.6431.
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Li, H;
Zhang, Z;
Godakanda, VU;
Chiu, Y-J;
Angkawinitwong, U;
Patel, K;
Stapleton, PG;
... Williams, GR; + view all
(2019)
The effect of collection substrate on electrospun ciprofloxacin-loaded poly(vinylpyrrolidone) and ethyl cellulose nanofibers as potential wound dressing materials.
Materials Science and Engineering: C
, 104
, Article 109917. 10.1016/j.msec.2019.109917.
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Lumlerdkij, N;
Boonrak, R;
Booranasubkajorn, S;
Akarasereenont, P;
Heinrich, M;
(2019)
In vitro protective effects of plants frequently used traditionally in cancer prevention in Thai traditional medicine: An ethnopharmacological study.
Journal of Ethnopharmacology
, 250
, Article 112409. 10.1016/j.jep.2019.112409.
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M
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Mack, AR;
Barnes, MD;
Taracila, MA;
Hujer, AM;
Hujer, KM;
Cabot, G;
Feldgarden, M;
... Bonomo, RA; + view all
(2019)
A standard numbering scheme for class C β-lactamases.
Antimicrobial Agents and Chemotherapy
10.1128/AAC.01841-19.
(In press).
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Mackonochie, M;
Heinrich, M;
(2019)
Materia medica chests: Investigating the 19th century use of botanicals by different medical professions.
Journal of Herbal Medicine
, 16
, Article 100255. 10.1016/j.hermed.2019.100255.
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Manukyan, A;
Lumlerdkij, N;
Heinrich, M;
(2019)
Caucasian endemic medicinal and nutraceutical plants: In vitro antioxidant and cytotoxic activities and bioactive compounds.
Journal of Pharmacy and Pharmacology
, 71
(7)
pp. 1152-1161.
10.1111/jphp.13093.
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Moore, BJR;
Islam, B;
Ward, S;
Jackson, O;
Armitage, R;
Blackburn, J;
Haider, S;
(2019)
Repurposing of Tranilast for Potential Neuropathic Pain Treatment by Inhibition of Sepiapterin Reductase in the BH₄ Pathway.
ACS Omega
, 4
(7)
pp. 11960-11972.
10.1021/acsomega.9b01228.
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O
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Oyedemi, BO;
Maria, KE;
Stapleton, PD;
Gibbons, S;
(2019)
Capsaicin and gingerol analogues inhibit the growth of efflux-multidrug resistant bacteria and R-plasmids conjugal transfer.
Journal of Ethnopharmacology
, 245
, Article 111871. 10.1016/j.jep.2019.111871.
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P
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Paredes, ME;
Morales, RE;
Lima, WK;
Hu, S;
Jurado, AL;
Farchi, E;
Prieto, JM;
(2019)
Morphoanatomical and phytochemical studies for the quality control of Neurolaena lobata (L.) R.Br. ex Cass. (Asteraceae).
Blacpma (Boletín Latinoamericano Y Del Caribe De Plantas Medicinales Y Aromáticas)
, 18
(3)
pp. 277-288.
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Penny, M;
Rao, Z;
Peniche, B;
Hilton, S;
(2019)
Modular 3D Printed Compressed Air Driven Continuous‐Flow Systems for Chemical Synthesis.
European Journal of Organic Chemistry
, 2019
(23)
pp. 3783-3787.
10.1002/ejoc.201900423.
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Pérez-Cantero, A;
Serrano, DR;
Navarro-Rodríguez, P;
Schätzlein, AG;
Uchegbu, IF;
Torrado, JJ;
Capilla, J;
(2019)
Increased Efficacy of Oral Fixed-Dose Combination of Amphotericin B and AHCC® Natural Adjuvant against Aspergillosis.
Pharmaceutics
, 11
(9)
, Article 456. 10.3390/pharmaceutics11090456.
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R
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Riccio, F;
Talapatra, SK;
Oxenford, S;
Angell, R;
Mazzon, M;
Kozielski, F;
(2019)
Development and validation of RdRp Screen, a crystallization screen for viral RNA-dependent RNA polymerases.
Biology Open
, 8
, Article bio037663. 10.1242/bio.037663.
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Romero, R;
Ramanathan, A;
Yuen, T;
Bhowmik, D;
Mathew, M;
Munshi, LB;
Javaid, S;
... Zaidi, M; + view all
(2019)
Mechanism of glucocerebrosidase activation and dysfunction in Gaucher disease unraveled by molecular dynamics and deep learning.
Proceedings of the National Academy of Sciences of the United States of America
10.1073/pnas.1818411116.
(In press).
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S
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Scotti, F;
Lobel, K;
Booker, A;
Heinrich, M;
(2019)
St. John's Wort (Hypericum perforatum) Products - How Variable Is the Primary Material?
Frontiers in Plant Science
, 9
, Article 1973. 10.3389/fpls.2018.01973.
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Smart, TG;
Stephenson, FA;
(2019)
A half century of γ-aminobutyric acid.
Brain and Neuroscience Advances
, 3
pp. 1-9.
10.1177/2398212819858249.
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Soumyanarayanan, U;
Ramanujulu, PM;
Mustafa, N;
Haider, S;
Fang Nee, AH;
Tong, JX;
Tan, KSW;
... Dymock, BW; + view all
(2019)
Discovery of a potent histone deacetylase (HDAC) 3/6 selective dual inhibitor.
European Journal of Medicinal Chemistry
, 184
, Article 111755. 10.1016/j.ejmech.2019.111755.
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Stowe, CL;
Burley, TA;
Allan, H;
Vinci, M;
Kramer-Marek, G;
Ciobota, DM;
Parkinson, GN;
... Pule, MA; + view all
(2019)
Near-infrared dual bioluminescence imaging in mouse models of cancer using infraluciferin.
eLife
, 8
, Article e45801. 10.7554/eLife.45801.
(In press).
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T
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Taylor, SE;
O'Connor, CM;
Wang, Z;
Shen, G;
Song, H;
Leonard, D;
Sangodkar, J;
... Narla, G; + view all
(2019)
The highly recurrent PP2A Aα-subunit mutation P179R alters protein structure and impairs PP2A enzyme function to promote endometrial tumorigenesis.
Cancer Research
, 79
(16)
pp. 4242-4257.
10.1158/0008-5472.CAN-19-0218.
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Timberlake, AT;
Jin, SC;
Nelson-Williams, C;
Wu, R;
Furey, CG;
Islam, B;
Haider, S;
... Lifton, RP; + view all
(2019)
Mutations in TFAP2B and previously unimplicated genes of the BMP, Wnt, and Hedgehog pathways in syndromic craniosynostosis.
Proceedings of the National Academy of Sciences of the United States of America
, 116
(30)
pp. 15116-15121.
10.1073/pnas.1902041116.
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Todd, MH;
(2019)
Six Laws of Open Source Drug Discovery.
ChemMedChem
, 14
(21)
pp. 1804-1809.
10.1002/cmdc.201900565.
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Tse, EG;
Korsik, M;
Todd, MH;
(2019)
The past, present and future of anti-malarial medicines.
Malaria Journal
, 18
(1)
, Article 93. 10.1186/s12936-019-2724-z.
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U
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Uchegbu, I;
Wang, Z;
Xiong, G;
Tsang, A;
Schatzlein, A;
(2019)
Nose to brain delivery.
Journal of Pharmacology and Experimental Therapeutics
, 370
(3)
pp. 593-601.
10.1124/jpet.119.258152.
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V
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Van Melis, CGW;
Penny, MR;
Garcia, AD;
Petti, A;
Dobbs, AP;
Hilton, ST;
Lam, K;
(2019)
Supporting-Electrolyte-Free Electrochemical Methoxymethylation of Alcohols Using a 3D-Printed Electrosynthesis Continuous Flow Cell System.
ChemElectroChem
, 6
(16)
pp. 4144-4148.
10.1002/celc.201900815.
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Vasu, D;
de Arriba, ALF;
Leitch, JA;
de Gombert, A;
Dixon, DJ;
(2019)
Primary alpha-tertiary amine synthesis via alpha-C-H functionalization.
Chemical Science
, 10
(11)
pp. 3401-3407.
10.1039/c8sc05164j.
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W
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Welker Leng, KR;
Castañeda, CA;
Decroos, C;
Islam, B;
Haider, SM;
Christianson, DW;
Fierke, CA;
(2019)
Phosphorylation of Histone Deacetylase 8: Structural and Mechanistic Analysis of the Phosphomimetic S39E Mutant.
Biochemistry
, 58
(45)
pp. 4480-4493.
10.1021/acs.biochem.9b00653.
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Y
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Yeung, AWK;
Tzvetkov, NT;
Gupta, VK;
Gupta, SC;
Orive, G;
Bonn, GK;
Fiebich, B;
... Atanasov, AG; + view all
(2019)
Current research in biotechnology: Exploring the biotech forefront.
Current Research in Biotechnology
, 1
pp. 34-40.
10.1016/j.crbiot.2019.08.003.
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Z
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Zhai, Q;
Gao, C;
Ding, J;
Zhang, Y;
Islam, B;
Lan, W;
Hou, H;
... Wei, D; + view all
(2019)
Selective recognition of c-MYC Pu22 G-quadruplex by a fluorescent probe.
Nucleic Acids Research
, 47
(5)
pp. 2190-2204.
10.1093/nar/gkz059.
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Zhang, Y;
Kung, C-P;
Sil, BC;
Lane, ME;
Hadgraft, J;
Heinrich, M;
Sinko, B;
(2019)
Topical Delivery of Niacinamide: Influence of Binary and Ternary Solvent Systems.
Pharmaceutics
, 11
(12)
, Article 668. 10.3390/pharmaceutics11120668.
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Zhang, Y;
Lane, M;
Hadgraft, J;
Heinrich, M;
Chen, T;
Lian, G;
Sinko, B;
(2019)
A comparison of the in vitro permeation of niacinamide in mammalian skin and in the Parallel Artificial Membrane Permeation Assay (PAMPA) model.
International Journal of Pharmaceutics
, 556
pp. 142-149.
10.1016/j.ijpharm.2018.11.065.
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Zhang, Y;
Sil, BC;
Kung, C-P;
Hadgraft, J;
Heinrich, M;
Sinko, B;
Lane, ME;
(2019)
Characterization and topical delivery of phenylethyl resorcinol.
International Journal of Cosmetic Science
, 41
(5)
pp. 479-488.
10.1111/ics.12565.
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