eprintid: 10203576
rev_number: 7
eprint_status: archive
userid: 699
dir: disk0/10/20/35/76
datestamp: 2025-01-20 11:03:56
lastmod: 2025-01-20 11:03:56
status_changed: 2025-01-20 11:03:56
type: article
metadata_visibility: show
sword_depositor: 699
creators_name: Yeung, Charlotte
creators_name: Mccoubrey, Laura E
creators_name: Basit, Abdul W
title: Advances in colon-targeted drug technologies
ispublished: pub
divisions: UCL
divisions: B02
divisions: C08
divisions: D10
divisions: G08
keywords: Artificial intelligence and machine learning, colonic targeting, gastro-resistant film coatings, mesalamine
formulations, oral drug delivery systems and the large intestine
note: This is an open access article distributed under the Creative Commons
Attribution License 4.0 (CCBY), which permits unrestricted use, distribution, and reproduction in any medium, provided the original work is
properly cited.
abstract: PURPOSE OF REVIEW: 
Herein, we present an overview of innovative oral technologies utilized in colonic drug delivery systems
that have made significant translational and clinical advancements to treat inflammatory bowel disease
(IBD) in recent years.

RECENT FINDINGS: 
The colon is home to distinct physiological conditions, such as pH and microbiota, that have been
exploited in the development of colonic drug delivery systems for the treatment of local and systemic
diseases. However, given the intra and interindividual variability in the gastrointestinal tract of both healthy
and diseased states, various systems have shown inconsistencies in targeted drug release to the colon.
Recent breakthroughs have led to systems that incorporate multiple independent trigger mechanisms,
ensuring drug release even if one mechanism fails due to physiological variability. Such advanced
platforms have bolstered the development of oral biologics delivery, an especially promising direction
given the lack of commercially available oral antibody medications for IBD. These concepts can be further
enhanced by employing 3D printing which enables the personalisation of medicines.

SUMMARY: 
Leveraging these novel technologies can accurately deliver therapeutics to the colon, allowing for
treatments beyond gastrointestinal tract diseases. To realize the full potential of colonic drug delivery, it is
paramount that research focuses on the clinical translatability and scalability of novel concepts.
date: 2025-01
date_type: published
publisher: LIPPINCOTT WILLIAMS & WILKINS
official_url: https://doi.org/10.1097/mog.0000000000001064
oa_status: green
full_text_type: pub
language: eng
primo: open
primo_central: open_green
verified: verified_manual
elements_id: 2334277
doi: 10.1097/MOG.0000000000001064
medium: Print-Electronic
pii: 00001574-202501000-00004
lyricists_name: Basit, Abdul
lyricists_id: ABASI56
actors_name: Gaisford, Simon
actors_name: Harris, Jean
actors_id: SGAIS88
actors_id: JAHAR68
actors_role: owner
actors_role: impersonator
full_text_status: public
publication: Current Opinion in Gastroenterology
volume: 41
number: 1
pagerange: 9-15
pages: 7
event_location: United States
issn: 0267-1379
citation:        Yeung, Charlotte;    Mccoubrey, Laura E;    Basit, Abdul W;      (2025)    Advances in colon-targeted drug technologies.                   Current Opinion in Gastroenterology , 41  (1)   pp. 9-15.    10.1097/MOG.0000000000001064 <https://doi.org/10.1097/MOG.0000000000001064>.       Green open access   
 
document_url: https://discovery.ucl.ac.uk/id/eprint/10203576/1/Advances%20in%20colon-targeted%20drug%20technologies.pdf