?url_ver=Z39.88-2004&rft_val_fmt=info%3Aofi%2Ffmt%3Akev%3Amtx%3Ajournal&rft.aulast=Woodward&rft.aufirst=HL&rft.au=Woodward%2C+HL&rft.title=Journal+of+Medicinal+Chemistry&rft.issn=1520-4804&rft.pages=8226-8240&rft.issue=18&rft.date=27+September+2018&rft.atitle=Introduction+of+a+Methyl+Group+Curbs+Metabolism+of+Pyrido%5B3%2C4-d%5Dpyrimidine+Monopolar+Spindle+1+(MPS1)+Inhibitors+and+Enables+the+Discovery+of+the+Phase+1+Clinical+Candidate+N2-(2-Ethoxy-4-(4-methyl-4H-1%2C2%2C4-triazol-3-yl)phenyl)-6-methyl-N8-neopentylpyrido%5B3%2C4-d%5Dpyrimidine-2%2C8-diamine+(BOS172722)&rft.volume=61&rft.genre=article